Medicinal Chemistry and Drug Design

Maynooth University

Course Description

  • Course Name

    Medicinal Chemistry and Drug Design

  • Host University

    Maynooth University

  • Location

    Dublin, Ireland

  • Area of Study

    Chemistry, Pharmacy

  • Language Level

    Taught In English

  • Prerequisites

    CH307, CH308, CH309, CH310

  • Course Level Recommendations

    Upper

    ISA offers course level recommendations in an effort to facilitate the determination of course levels by credential evaluators.We advice each institution to have their own credentials evaluator make the final decision regrading course levels.

    Hours & Credits

  • ECTS Credits

    5
  • Recommended U.S. Semester Credits
    2
  • Recommended U.S. Quarter Units
    3
  • Overview

    Medicinal Chemistry, Computational Drug Design, Heterocyclic Drugs

    This module provides an introduction to important concepts in medicinal chemistry, computational drug design and heterocyclic drugs:

    (i) Medicinal Chemistry. Material covered includes the purpose and principles of medicinal chemistry in the drug discovery, design and development process, pharmacodynamic and pharmacokinetic aspects of drug action in the context of chemical structure, structure-activity relationships for optimization of lead compounds and sources and approaches to the discovery of lead compounds.

    (ii) Introduction to computational drug design. Material covered includes structure and ligand based techniques for hit compound discovery and hit-to-lead optimization, molecular modelling, pharmacophore and chemoinformatics in drug design.

    (ii) Heterocyclic drugs. Material covered includes an introduction to the different types of heterocycles found in nature and as part of drugs and their physicochemical characteristics and mechanism of action of heterocyclic drugs such as antibiotics, antiviral drugs, anticancer agents and heterocyclic drugs acting in CNS and in heart disease.

Course Disclaimer

Courses and course hours of instruction are subject to change.

Credits earned vary according to the policies of the students' home institutions. According to ISA policy and possible visa requirements, students must maintain full-time enrollment status, as determined by their home institutions, for the duration of the program.

ECTS (European Credit Transfer and Accumulation System) credits are converted to semester credits/quarter units differently among U.S. universities. Students should confirm the conversion scale used at their home university when determining credit transfer.

Please reference fall and spring course lists as not all courses are taught during both semesters.

Please note that some courses with locals have recommended prerequisite courses. It is the student's responsibility to consult any recommended prerequisites prior to enrolling in their course.